2-(1-Piperidinyl)-1,3-benzothiazole

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چکیده

منابع مشابه

Photoinduced proton coupled electron transfer in 2-(2'-hydroxyphenyl)-benzothiazole.

We characterize the structural and electronic changes during the photoinduced enol-keto tautomerization of 2-(2'-hydroxyphenyl)-benzothiazole (HBT) in a nonpolar solvent (tetrachloroethene). We quantify the redistribution of electronic charge and intramolecular proton translocation in real time by combining UV-pump/IR-probe spectroscopy and quantum chemical modeling. We find that the photophysi...

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Synthesis, Characterization and Antimicrobial activity of 2- Amino-1,3-benzothiazole, Schiff bases and Azo dyes of 2-Amino- 1,3-benzothiazole

2-Amino-1,3-benzothiazole was synthesized and schiff bases were prepared by reacting a series of aromatic aldehydes with 2-amino-1,3-benzothiazole to form a number of potentially biologically active compounds. Azo dyes of 2-amino-1,3-benzothiazole were synthesized by reacting various aromatic amines , substituted amines and phenols. The structures of 2-amino-1,3-benzothiazole, Schiff bases and ...

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[ D - Ala 2 , ( Fs ) Phe 4 ] - Dynorphin 1 - - 13 - N H 2 ( DAFPHEDYN ) : A Potent Analog of Dynorphin 1 - 13

WALKER, J. M., D. H. COY, E. A. YOUNG, G. BALDRIGHI, S. F. SIEGEL, W. D. BOWEN AND H. AKIL. [D-AIa z, (F~)Phe4]-Dynorphin~_la-NH2 (DAFPHEDYN): A potent analog of dynorphin 1-13. PEPTIDES 8(5) 811-817, 1987.-Intracerebroventricular administration of the dynorphin analog, [D-Ala2,(Fs)Phe4]-dynorphint_l~-NH2 (DAFPHEDYN) in rats produced diuresis and profound analgesia. Both effects were antagonize...

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Mechanism-based inactivation of cytochromes P450 2B1 and P450 2B6 by 2-phenyl-2-(1-piperidinyl)propane.

2-Phenyl-2-(1-piperidinyl)propane (PPP), an analog of phencyclidine, was tested for its ability to inactivate cytochrome P450s (P450s) 2B1 and 2B6. PPP inactivated the 7-(benzyloxy)resorufin O-dealkylation activity of liver microsomes obtained from phenobarbital-induced rats with a K(I) of 11 microM. The 7-ethoxy-4-(trifluoromethyl)coumarin O-deethylation activity of purified rat liver P450 2B1...

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Interaction of [2-(alkyloxy)-phenyl]-2-(1-piperidinyl)ethyl esters of carbamic acid with dipalmitoylphosphatidylglycerol model membranes: a calorimetric study.

As detected by adiabatic differential scanning microcalorimetry, [2-(alkyloxy)-phenyl]-2-(1-piperidinyl)ethyl esters of carbamic acid (CnPPEECA, n is the number of carbon atoms in the alkyloxy substituent) with local anesthetic and antiarrhythmic activities interact with 1,2-dipalmitoyl-sn-glycero-3-[phosphorac-(1-glycerol)] model membranes (DPPG). CnPPEECAs form solid-like solutions with DPPG ...

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ژورنال

عنوان ژورنال: Acta Crystallographica Section E Structure Reports Online

سال: 2005

ISSN: 1600-5368

DOI: 10.1107/s160053680500320x